Phase II metabolism (conjugation reactions) — Flashcards

Phase II metabolism (conjugation reactions) — Flashcards

Phase II metabolism (conjugation reactions) — Flashcards
#1

Isoniazid is metabolized by the hepatic enzyme _____

#2

Azathioprine and 6-mercaptopurine are metabolized by _____ (enzyme)

#3

What phase of drug metabolism includes methylation, glucuronidation, acetylation, and sulfation (i.e. conjugation)? _____

#4

Isoniazid hepatotoxicity results in an asymptomatic rise in _____ on LFTs

#5

What toxic intermediate is formed in small amounts by metabolism of acetaminophen? _____

#6

_____ toxicity is associated with Isoniazid use

Want unlimited flashcards?

Get full access to all flashcards, spaced repetition, and progress tracking.

Start For Free