Phase I metabolism (oxidation, reduction, hydrolysis) — Flashcards

Phase I metabolism (oxidation, reduction, hydrolysis) — Flashcards

Phase I metabolism (oxidation, reduction, hydrolysis) — Flashcards
#1

Which one of the following drugs is a cytochrome p450 inducer?_____

#2

Phenobarbital is an _____ of CYP-450

#3

Rifabutin _____ cytochrome p450 (induces or inhibits)

#4

Azoles _____ cytochrome p450

#5

Phase _____ drug metabolism usually yields slightly polar, water-soluble metabolites (often still active)

#6

What phase of drug metabolism includes reduction, oxidation, and hydrolysis? _____

#7

Theophylline is metabolized by _____

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